Mechanistic investigation of aziridine aldehyde-driven peptide macrocyclization: the imidoanhydride pathway

نویسندگان

  • Serge Zaretsky
  • Jennifer L. Hickey
  • Joanne Tan
  • Dmitry Pichugin
  • Benjamin K. W. Chung
  • Conor C. G. Scully
  • Andrei K. Yudin
چکیده

Davenport Research Laboratories, Departme St. George Street, Toronto, Ontario M5S utoronto.ca Encycle Therapeutics Inc., 101 College Stre Canada Center for Structural Investigations of Co Department of Chemistry, University of T Ontario M5S 3H6, Canada † Electronic supplementary information ( and characterization data. CCDC 14 crystallographic data in CIF or o 10.1039/c5sc01958c Cite this: Chem. Sci., 2015, 6, 5446

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تاریخ انتشار 2015